PUBLICATIONS

2009-2005

Novel Inhibitors of Fatty Acid Synthase with Anticancer Activity

T. Puig, C. Turrado, B. Benhamú, H. Aguilar, J. Relat, S. Ortega-Gutiérrez, G. Casals, P.F. Marrero, A. Urruticoechea, D. Haro, M.L. López-Rodríguez, R. Colomer

Synthesis of new serotonin 5-HT7 receptor ligands. Determinants of 5-HT7/5-HT1A receptor selectivity

R.A. Medina, J. Sallander, B. Benhamú, E. Porras, M. Campillo, L. Pardo, M.L. López-Rodríguez

Central nervous system (CNS)-related pathologies

M.L. López-Rodríguez

Targeted disruption of the PME-1 gene causes loss of demethylated PP2A and perinatal lethality in mice

S. Ortega-Gutiérrez, D. Leung, S. Ficarro, E.C. Peters, B.F. Cravatt

The medicinal chemistry of agents targeting monoacylglycerol lipase

A. Viso, J.A. Cisneros, S. Ortega-Gutiérrez

Structure-activity relationship of a series of inhibitors of monoacylglycerol hydrolysis--comparison with effects upon fatty acid amide hydrolase

J.A. Cisneros, S. Vandevoorde, S. Ortega-Gutiérrez, C. Paris, C.J. Fowler, M.L. López-Rodríguez

Structural models of class a G protein-coupled receptors as a tool for drug design: insights on transmembrane bundle plasticity

X. Deupi, N. Dölker, M.L. López-Rodríguez, M. Campillo, J.A. Ballesteros, L. Pardo

Identification of a novel endocannabinoid-hydrolyzing enzyme expressed by microglial cells

G.G. Muccioli, C. Xu, E. Odah, E. Cudaback, J.A. Cisneros, D.M. Lambert, M.L. López Rodríguez, S. Bajjalieh, N. Stella

Neurochemical effects of the endocannabinoid uptake inhibitor UCM707 in various rat brain regions

E. de Lago, S. Ortega-Gutiérrez, J.A. Ramos, M.L. López Rodríguez, J. Fernández-Ruiz

The role of internal water molecules in the structure and function of the rhodopsin family of G protein-coupled receptors

L. Pardo, X. Deupi, N. Dölker, M.L. López-Rodríguez, M. Campillo

Synthesis of highly substituted enantiopure piperazines and ketopiperazines from vicinal N-sulfinyl diamines

A. Viso, R. Fernández de la Pradilla, A. Flores, A. García, M. Tortosa, M.L. López-Rodríguez

CB1 and CB2 cannabinoid receptor binding studies based on modeling and mutagenesis approaches

S. Ortega-Gutiérrez, M.L. López-Rodríguez

Cannabinoids

M.L. López-Rodríguez

A three-dimensional pharmacophore model for 5-hydroxytryptamine6 (5-HT6) receptor antagonists.

M.L. López-Rodríguez, B. Benhamú, T. de la Fuente, A. Sanz, L. Pardo, M. Campillo

Activation of the endocannabinoid system as therapeutic approach in a murine model of multiple sclerosis.

S. Ortega-Gutiérrez, E. Molina-Holgado, A. Arévalo-Martín, F. Correa, A. Viso, M.L. López-Rodríguez, V. Di Marzo, C. Guaza

Synthesis and structure-activity relationships of a new model of arylpiperazines. 8. Computational simulation of ligand-receptor interaction of 5-HT(1A)R agonists with selectivity over alpha1-adrenoceptors

M.L. López-Rodríguez, M.J. Morcillo, E. Fernández, B. Benhamú, I. Tejada, D. Ayala, A. Viso, M. Campillo, L. Pardo, M. Delgado, J. Manzanares, J.A. Fuentes.

Anxiolytic-like effect of a serotonergic ligand with high affinity for 5-HT1A, 5-HT2A and 5-HT3 receptors

M. Delgado, A.G. Caicoya, V. Greciano, B. Benhamú, M.L. López-Rodríguez, M.S. Fernández-Alfonso, M.A. Pozo, J. Manzanares, J.A. Fuentes

Involvement of cannabinoids in cellular proliferation

M.L. López-Rodríguez, A. Viso, S. Ortega-Gutiérrez, I. Díaz-Laviada

Therapeutic perspectives of inhibitors of endocannabinoid degradation

S. Ortega-Gutiérrez

Effect of repeated systemic administration of selective inhibitors of endocannabinoid inactivation on rat brain endocannabinoid levels

E. de Lago, S. Petrosino, M. Valenti, E. Morera, S. Ortega-Gutiérrez, J. Fernandez-Ruiz, V. Di Marzo

Effect of anandamide uptake inhibition in the production of nitric oxide and in the release of cytokines in astrocyte cultures

S. Ortega-Gutiérrez, E. Molina-Holgado, C. Guaza